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1 Aug. THE JAPANESE JOURNAL OF ANTIBIOTICS ( 15 ) 1. MDS collagenase /

2 390( 16 ) THE JAPANESE JOURNAL OF ANTIBIOTICS 58 4 Aug NTT

3 Aug. THE JAPANESE JOURNAL OF ANTIBIOTICS ( 17 ) 1 MDS collagenase Matrix metalloproteinases (MMP)-2, MMP-9 IV collagenase MMP-2, MMP-8, MMP-9 (Myelodysplastic syndrome: MDS) collagenase MDS collagenase Collagenase MDS collagenase MDS FAB RA (refractory anemia) 31 RARS (refractory anemia with ringed sideroblast) 4 RAEB (refractory anemia with excess of blasts) 5 RAEBt (refractory anemia with excess of blasts in transformation) 1 CMML (chronic myelomonocytic leukemia) 2 post-mds AML (acute myeloid leukemia) 2 5 collagenase CellProbe (Beckman Coulter, Fullerton, CA, USA) CellProbe MMP-2, MMP-8, MMP-9 II IV collagenase CellProbe collagenase collagenase CellProbe collagenase MDS collagenase MDS collagenase (p 0.05) FAB (Table 1) Table 1. Collagenase

4 392( 18 ) THE JAPANESE JOURNAL OF ANTIBIOTICS 58 4 Aug. IPSS (International Prognostic Scoring System) collagenase (Table 2) MDS NAP (Neutrophil Alkalyne Phosphatase Score) NAP collagenase (Table 3) collagenase MDS collagenase MDS 1,000/ml 37.5 C 7 MDS 50 6 collagenase (p 0.01) MDS ( p 0.01) (Table 4) collagenase (SD) (p ) Collagenase (Table 5) 1 Table 2. IPSS collagenase Table 3. NAP collagenase Table 4. collagenase Table 5. Collagenase *

5 Aug. MDS collagenase MDS collagenase collagenase MDS collagenase NAP collagenase THE JAPANESE JOURNAL OF ANTIBIOTICS ( 19 ) NAP G-CSF G-CSF G-CSF collagenase collagenase collagenase 6

6 394( 20 ) THE JAPANESE JOURNAL OF ANTIBIOTICS 58 4 Aug ) 2) 1) 1) 2) C / 9 730/ml 510/m l 210/m l 10/ml / ml 5.8g/dl 17.3% 6,600/ml 6.3 /ml CRP 5.27mg/dl M/E % (Myelodysplastic syndrome: MDS) CD4 53.4% (32 48), CD8 32.2% (21 33) PHA 956 cpm (26,000 53,000), ConA 1,230 cpm (20,000 48,000) Gaffky Mycobacterium avium 3 3mm G-CSF ciclosporin (CyA) (Fig. 1) M. avium isoniazid (INH), ethambutol (EB) CRP rifampicin (RFP), clarithromycin (CAM) CRP 1.20 mg/dl ciclosporin ethambutol, clarithromycin ciclosporin, ethambutol, clarithromycin cm (Fig. 2) 10

7 Aug. THE JAPANESE JOURNAL OF ANTIBIOTICS ( 21 ) Fig. 1. Fig MRI L2 T2 L4 (Fig. 3) 3,950/m l 3,349/ml

8 396( 22 ) THE JAPANESE JOURNAL OF ANTIBIOTICS 58 4 Aug. Fig. 3. MRI Fig. 4. MRI Cryptococcus neoformans ( ) Fluconazole (FLCZ) 200 mg/ CRP 2.81 mg/dl MRI L2 L4 (Fig. 4) Fluconazole 200 mg /m l 20/m l 9.6 g/ dl CRP 4.91 mg/dl MRI

9 Aug. Cryptococcus neoformans THE JAPANESE JOURNAL OF ANTIBIOTICS ( 23 )

10 398( 24 ) THE JAPANESE JOURNAL OF ANTIBIOTICS 58 4 Aug. 3 Fluconazole (FLCZ) (ITCZ) FLCZ ITCZ FLCZ FLCZ ITCZ 4 FLCZ mg/ ITCZ 200 mg/ 100 mg/ (None) 181 FLCZ (FLCZ) 71 ITCZ (ITCZ) 91 FLCZ ITCZ (FLCZÆITCZ) 8 ITCZ FLCZ (ITCZÆFLCZ) (Table 1) (Fig. 1) FLCZ 27.9 ITCZ % (10/71) ITCZ 4.4% (4/91) (Table 1) ITCZ ITCZ FLCZ p 0.01: c 2 ITCZ FLCZ FLCZ ITCZ FLCZ 1

11 Aug. THE JAPANESE JOURNAL OF ANTIBIOTICS ( 25 ) Table 1. Fig. 1. (non-hodgkin s lymphoma: NHL) 98 (acute myeloid leukemia: AML) 67 (acute lymphoblastic leukemia: ALL) 20 (multiple myeloma: MM) 15 (Table 2) ITCZ 0% (0/34) FLCZ 19.4% (7/ 36) p 0.02: c 2 ITCZ FLCZ p 0.004: c 2

12 400( 26 ) THE JAPANESE JOURNAL OF ANTIBIOTICS 58 4 Aug. Table 2. Table 3.

13 Aug. THE JAPANESE JOURNAL OF ANTIBIOTICS ( 27 ) Table (Table 3) p 0.009: c 2 FLCZ AMPH-B ITCZ 3.3% (3/91) ITCZ FLCZ 16.1% p 0.01: c 2 (Table 4) FLCZ ITCZ ITCZ FLCZ ITCZ b-d-

14 402( 28 ) THE JAPANESE JOURNAL OF ANTIBIOTICS 58 4 Aug. 4 / Fluconazole (FLCZ) (ITCZ) Fluconazole (oral solution) Fluconazole 500/ml Fluconazole 200 mg/ 1 1 H 2 Fluconazole 1,000/ml 7 B 300 mg/ b -D- 1,000/ml 7 Fluconazole 14 (Table 1) 14 4 (28.6%)

15 Aug. THE JAPANESE JOURNAL OF ANTIBIOTICS ( 29 ) Table 1. Table 2. Fig. 1. Fluconazole 14 5 (35.7%) (Table 2) Fluconazole 2 (possible) /ml CT Micafungin 250 ng/ml 500 ng/ml 250 ng/ml (Fig. 1) (OH- ITCZ) Fig. 2.

16 404( 30 ) THE JAPANESE JOURNAL OF ANTIBIOTICS 58 4 Aug. (Fig. 2) Fluconazole 200 mg/ Fluconazole MIC ng/ml 1) ng/ml 2), 500 ng/ml 3) 250 ng/ml Fluconazole in vitro (OH-ITCZ) 14 Fluconazole 2 b-d- 2 b-d- Fluconazole Fluconazole 1 1) BOOGAERTS, M. A., et al.: Mycoses, ) BOYLE, B. M., et al.: Transplant Infection Disease, ) GLASMACHER, A., et al.: Mycoses, 1999

051

051 June THE JAPANESE JOURNAL OF ANTIBIOTICS 57 3 295( 83 ) NTT 1. 2. 3. 4. CHOP-R 5. DNA 1 296( 84 ) THE JAPANESE JOURNAL OF ANTIBIOTICS 57 3 June 3 1 2003 10 4 1 NTT June THE JAPANESE JOURNAL OF ANTIBIOTICS

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