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1 I ab c AMPcAMP a b c camp camp Ca 2+ β1 camp A camp camp A β1 p.156 β p.146 b. p.157 p135 (ANP) p157 c PDE-III p.157 p.157, 183 PDE C Ca PDE-III Ia Na + p.161 ACE p a b c d --- Na ß Ca K e --- Na + K + -ATPase ---
2 1abc2abe3ade4bcd5cde a. (p.161)ib Na+ (p.119) b. (p.163)ii β c. (p.163) Ca IV d. (p.163)k + III e. (p.163, p.152) Na + /K + -ATPase Ca 2+ a b c d e 133 a Na + K + b Na + cd- Na + d K + 1ab2ac3ad4bc5bd6cd a. (p.176) Na + /Cl - b. Na + (p.177) c. D- (p.178) Na + d. (p.178) Na + Na+ K + K al- -S-S- b c d ß2 e d a. L- (p.188) SS b. (p.188) c. (p.189) d. (p.185) β2 β1 e. (p.87)
3 187 a b ACE c ACE II d II II e ß 1abc2abe3acd4bde5cde a. II NaCl K + b. ACE ACE ACE ACE c. p ACE II d. II II II ACE e. β (p.148) / a bna + Ia c dna + Ib e 1abd2abe3acd4bce5cde a. β (p.156) p II β III K+ IV Ca I Ia Ib bce ST-T a ß b c ß dca 2+ e 1abc2abe3acd4bde5cde p.133 p ST-T p.135p.141 cde
4 / 198/100 mmhg K + a ß bca 2+ c d ACE e II 1abc2abe3acd4bde5cde p Ca 2+ ACE II ACE II II K+ K + bde 193 a b c d e d a. b. c. (p.188) d. e. 194 a b ß2 c d e 1abe2acd3ace4bcd5bde
5 a. (COPD) b. 2 Gs camp Ca 2+ camp Ca 2+ c. d. e. COPD ace a b c d ( ) e 1(abc)2(abe)3(acd)4(bde)5(cde) a. b. c. d. e. acd a b c d e ---- ß Gs ---- M C ---- GABAA ---- Cl HT Gi (ab)2(ad)3(bc)4(ce)5(de) a. Gs camp b. M3 Gq C c. GABAA GABAA Cl - d. e. - ab
6 123 - B C B C 10 B C BC H1 H1 H2 (p.66)ssri PDE 132 ah +,K + -ATPase Na + Ca 2+ b c d e 1(ab)2(ae)3(bc)4(cd)5(de) a. Na + /K + -ATPase b. c. d, e. d, e de
7 a ß2 b c d e 1(abc)2(abe)3(ade)4(bcd)5(cde) 1 p.106, p. 137, p.146, p.163 a. b c d a b c D1 d 1(ab)2(ad)3(bc)4(bd)5(cd) a b cna + -K + -2Cl - d e 1(abc)2(abe)3(acd)4(bde)5(cde) a b AMP (camp) c ß2 ß1 d A2 e 1(abc)2(ace)3(ade)4(bcd)5(bde) mg/ 40 mg/ ST K + a b (ACE) c ß d 1(ab)2(ac)3(ad)4(bd)5(cd)
8 / 180/100 mmhg, a b Ca 2+ c ß d a1 e II 1(abc)2(abd)3(ace)4(bde)5(cde) a b c ß2 d 1(ab)2(ac)3(bc)4(bd)5(cd) aca 2+ b c d e GLP GLP 123 -
9 ) Ca 2 ß1 II a1
10 134 Na K + -ATPase Ca 2 camp ß1 Gi a 135 I2 136 ß K + Ca 2 Na ß ß2 L-
11 GFJ GFJ CYP3A4 GFJ GFJ GFJ Cmax GFJ 3 AMPcAMP ß Ca K +
12 ß Na + QT ß1 Ca 2+ D- II Cockcroft-Gault
13 ß ST ß CO2 O2 ß2 (NSAID) A B
14 a pd2 6.O7.O b A c A pa2 8.0 d B pa2 7.0 e M A 10-8 M 90% 1(a, b, c) 2 (a, b, e) 3(a, c, d)4(b, d, e) 5 (c, d, e) a ß1 b ß1 c a1 d a1 a2 a2 e aß 1(a, b)2(a, d)3(b, e)4(c, d)5(c, e) a b c d e AMP(cAMP) 1(a, c)2(a, d)3(b, d)4(b, e)5(c, e) Ca2+ a L Ca2+ b c d e 1(a, b, c) 2 (a, b, e) 3(a, c, d)4(b, d, e) 5 (c, d, e) a +
15 b Na + - K + c H + - K + d Na + - K + -2Cl - e Na + K + 1(a, b)2(a, d)3(b, c)4(c, e)5(d, e) a b c d e T 1(a, b)2(a, e)3(b, c)4(c, d)5(d, e) a b 5 c Ca 2+ d ß 1(a, b)2(a, c) 3(a, d)4(b, c)5(b, d) 6(c, d) a b a c ß d Ca e Na + K + 1(a, b,c) 2 (a, b, e) 3(a, c, d)4(a, d,e) 5 (b, c,d) 6(c, d, e) A-D 1 2 a A intrinsic activity1 b B A1/ c0.5
16 d100µm B 30µM e100µm B D a b c d e 1abc 2abe3ade 4bcd 5cde a100 b c d ST T a a b c d a e -----a a a1 b a2 c ß1 dß1
17 e ß2 1ab2ae3bc4cd5de a b c d e ab2ad3bc4ce5de a K b c a dß e 1ab2ad3be4cd5ce a b c d e Na Cl - 1ab2ae3bc4cd5de ae aa bbd cc B dba ec 1abd2a cd3 ace 4bce5bde a b IgE
18 c d e a b c 1 10 L d Vaughan Williams ana Ia b Ib Ic cß II I dk III eca 2 IV a GFR b Na K c Na d e 1ac2ae3bd4be5cd a b c d
19 mmhg 140 mgdlna 145 meqlk 3.8 meq LCl 104 meql OHCS6.5 mg 38 mg CT 131 I-metaiodobenzylguanidineMIBG a ß ß2 7 G G ADP G ADP GTPase G camp IP ac2ae3bd4be5cd II v I II 1ac2ae3bd4be5cd 137 ß1 a1 M1 NN
20 ß ß2 a1 191 ST ß mg mgday 3 QT 580 msec 67min torsades de pointes 2 3 QT QT
21 CYPIA2 CYPIA2 CYPIA2 CYP2D6 CYP2D6 CYP2D6 CYP3A4 CYP3A4 CYP3A4 207 ß- TDM 20 µgml 1abc2abd3ace 4bcd5bce6cde
A(6, 13) B(1, 1) 65 y C 2 A(2, 1) B( 3, 2) C 66 x + 2y 1 = 0 2 A(1, 1) B(3, 0) P 67 3 A(3, 3) B(1, 2) C(4, 0) (1) ABC G (2) 3 A B C P 6
1 1 1.1 64 A6, 1) B1, 1) 65 C A, 1) B, ) C 66 + 1 = 0 A1, 1) B, 0) P 67 A, ) B1, ) C4, 0) 1) ABC G ) A B C P 64 A 1, 1) B, ) AB AB = 1) + 1) A 1, 1) 1 B, ) 1 65 66 65 C0, k) 66 1 p, p) 1 1 A B AB A 67
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