日本化学療法学会雑誌第61巻第6号

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1 β Moraxella catarrhalis Escherichia coli Citrobacter Klebsiella pneumoniae Enterobacter cloacae Serratia marcescens Proteus Pseudomonas aeruginosa Acinetobacter Bacteroides fragilis β Haemophilus influenzae β H. influenzae β β E. coli K. pneumoniae Proteus mirabilis E. coli P. mirabilis β E. cloacae P. aeruginosa Acinetobacter S. marcescens P. aeruginosa P. mirabilis Proteus β H. influenzae H. influenzae

2 Key words β β β Pseudomonas aeruginosa β I Staphylococcus aureus Streptococcus pneumoniae S. pneumoniae Streptococcus Enterococcus faecalis Moraxella catarrhalis Escherichia coli Citrobacter Klebsiella pneumoniae Enterobacter cloacae Serratia marcescens Proteus mirabilis Proteus Providencia Haemophilus influenzae Acinetobacter Pseudomonas aeruginosa Bacteroides fragilis μ S. pneumoniae H. influenzae E. coli K. pneumoniae P. mirabilis μ μ S. pneumoniae H. influenzae S. pneumoniae

3 Table 1. Number of collected strains in items of clinical sources Total Blood % Expectoration No. of strains (%) % Urine % Pus % Spinal fluid % Others % Methicillin-susceptible Staphylococcus aureus Methicillin-susceptible coagulase-negative staphylococci S. pneumoniae Streptococcus species (other than S. pneumoniae) Enterococcus faecalis Moraxella catarrhalis Escherichia coli Citrobacter species Klebsiella pneumoniae Enterobacter cloacae Serratia marcescens Proteus mirabilis Indole-positive Proteus species Providencia species Haemophilus influenzae Pseudomonas aeruginosa Acinetobacter species Bacteroides fragilis group Total 4, , H. influenzae μ β μ B. fragilis μ μ S. pneumoniae H. influenzae β S. aureus μ μ S. pneumoniae μ S. pneumoniae μ μ S. pneumoniae μ S. pneumoniae H. influenzae β μ β H. influenzae P. aeruginosa μ μ μ P. aeruginosa β E. faecalis β β E. coli K. pneumoniae P. mirabilis P. aeruginosa E. cloacae S. marcescens Acinetobacter β β II β E. faecalis M. catarrhalis E. coli Citrobacter K. pneumoniae

4 Table 2. Number of -lactamase producing strains No. of strains No. of -lactamase producing strains % No. of ESBLs producing strains % No. of metallo- -lactamase producing strains Methicillin-susceptible Staphylococcus aureus Methicillin-susceptible coagulase-negative staphylococci Moraxella catarrhalis Escherichia coli Citrobacter species Klebsiella pneumoniae Enterobacter cloacae Serratia marcescens Proteus mirabilis Indole-positive Proteus species Providencia species Haemophilus influenzae Pseudomonas aeruginosa Acinetobacter species Bacteroides fragilis group Total 3,296 2, % E. cloacae S. marcescens Proteus P. aeruginosa Acinetobacter B. fragilis β E. coli β E. cloacae P. aeruginosa Acinetobacter S. pneumoniae E. faecalis M. catarrhalis μ E. coli E. coli E. coli E. coli Citrobacter K. pneumoniae E. cloacae S. marcescens P. mirabilis P. mirabilis Proteus Providencia H. influenzae β H. influenzae β H. influenzae β H. influenzae

5 Methicillin-susceptible Staphylococcus aureus (MSSA) Methicillin-susceptible coagulase-negative staphylococci (MSCNS) No. of strains Table 3. Susceptibilities of clinical isolates to antimicrobial agents tested Drug MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST 293 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX Streptococcus pneumoniae 267 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX Penicillin-susceptible Streptococcus pneumoniae (PSSP) Penicillin-intermediate Streptococcus pneumoniae (PISP) 112 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX (Continued)

6 Penicillin-resistant Streptococcus pneumoniae (PRSP) Streptococcus species (other than S. pneumoniae) No. of strains Drug Table 3. (Continued) MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST 62 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX Enterococcus faecalis 218 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX Moraxella catarrhalis 186 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX Escherichia coli 304 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX (Continued)

7 ESBLs producing Escherichia coli No. of strains Drug Table 3. (Continued) MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST 54 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX Citrobacter species 234 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX Klebsiella pneumoniae 231 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX Enterobacter cloacae 197 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX Serratia marcescens 249 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX (Continued) H. influenzae P. aeruginosa Acinetobacter

8 No. of strains Drug MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST Proteus mirabilis 218 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX Indole-positive Proteus species 114 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX Providencia species 80 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX Haemophilus influenzae 252 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX Lactamase-negative ampicillin-susceptible Haemophilus influenzae (BLNAS) Table 3. (Continued) 110 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX (Continued) B. fragilis III

9 -Lactamase-negative ampicillin-resistant Haemophilus influenzae (BLNAR) No. of strains Drug Table 3. (Continued) MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST 114 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM EM CPFX LVFX Pseudomonas aeruginosa 303 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX Acinetobacter species 240 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX Bacteroides fragilis group 185 TAZ/PIPC PIPC SBT/ABPC CAZ CFPM IPM/CS MEPM GM CPFX LVFX β β M. catarrhalis E. coli Citrobacter K. pneumoniae E. cloacae S. marcescens Proteus P. aeruginosa Acinetobacter B. fragilis E. coli Citrobacter K. pneumoniae E. cloacae S. marcescens P. aeruginosa B. fragilis β β H. influenzae β H. influenzae β β β H. influenzae β H. influenzae

10 β E. coli P. mirabilis P. aeruginosa P. mirabilis Proteus H. influenzae P. aeruginosa P. aeruginosa μ μ P. aeruginosa μ P. aeruginosa E. coli K. pneumoniae P. mirabilis μ H. influenzae H. influenzae μ μ S. pneumoniae μ μ μ

11 Pseudomonas aeruginosa β β β β Haemophilus influenzae β β Pseudomonas aeruginosa β bla Proteus mirabilis

12 β β Moraxella catarrhalis Escherichia coli Citrobacter Klebsiella pneumoniae Enterobacter cloacae Serratia marcescens Proteus Pseudomonas aeruginosa Acinetobacter Bacteroides fragilis Haemophilus influenzae β H. influenzae β E. coli, K. pneumoniae P. mirabilis E. coli, K. pneumoniae P. mirabilis β E. cloacae P. aeruginosa Acinetobacter S. marcescens P. aeruginosa S. aureus P. mirabilis Proteus Proteus mirabilis H. influenzae β H. influenzae Enterobacteriaceae

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