日本化学療法学会雑誌第64巻第4号

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1 β β Moraxella catarrhalisescherichia colicitrobacter Klebsiella pneumoniaeenterobacter cloacaeserratia marcescens Proteus Providencia Pseudomonas aeruginosaacinetobacter Bacteroides fragilis β β E. colik. pneumoniae P. mirabilis β P. aeruginosa Acinetobacter E. cloacae S. marcescens E. cloacae Staphylococcus aureus M catarrhalisp. mirabilis Proteus β Haemophilus influenzaeβ H. influenzae Streptococcus pneumoniae Streptococcus pneumoniae E.coli

2 Key words β β β I Staphylococcus aureus Streptococcus pneumoniaes. pneumoniae Streptococcus Enterococcus faecalismoraxella catarrhalisescherichia colicitrobacter Klebsiella pneumoniaeenterobacter cloacaeserratia marcescensproteus mirabilisproteus Providencia Haemophilus influenzaeacinetobacter Pseudomonas aeruginosa Bacteroides fragilis β μ S. pneumoniae H. influenzae E. colik. pneumoniae P. mirabilis μ μ S. pneumoniae H. in-

3 Table1.Number of collected in materials from clinical sources (%) Total Blood % Expectoration % Urine % Pus % Spinal fluid % Others % Methicillin-susceptible Staphylococcus aureus Methicillin-susceptible coagulase-negative staphylococci Streptococcus pneumoniae Streptococcus species (other than S. pneumoniae) Enterococcus faecalis Moraxella catarrhalis Escherichia coli Citrobacter species Klebsiella pneumoniae Enterobacter cloacae Serratia marcescens Proteus mirabilis Indole-positive Proteus species Providencia species Haemophilus influenzae Pseudomonas aeruginosa Acinetobacter species Bacteroides fragilis group Total 3, , ,

4 Table2.Number of -lactamase producing -lactamase producing % ESBLs producing % metallo- -lactamase producing Methicillin-susceptible Staphylococcus aureus Methicillin-susceptible coagulase-negative staphylococci Moraxella catarrhalis Escherichia coli Citrobacter species Klebsiella pneumoniae Enterobacter cloacae Serratia marcescens Proteus mirabilis Indole-positive Proteus species Providencia species Haemophilus influenzae Pseudomonas aeruginosa Acinetobacter species Bacteroides fragilis group Total 3,215 2, % fluenzae S. pneumoniae H. influenzae μ β μ B. fragilis μ μ S. pneumoniae H. influenzae β S. aureus μ μ S. pneumoniae μ S. pneumoniae Streptococcus pneumoniae μ μ S. pneumoniae Streptococcus pneumoniae μ S. pneumoniae Streptococcus pneumoniaeh. influenzae β μ β H. influenzae β β E. faecalis β β β β E. colik. pneumoniae P. mirabilis P. aeruginosae. cloacaes. marcescens Acinetobacter β β II β E. faecalis M. catarrhalise. colicitrobacter K. pneumoniaee. cloacaes. marcescens Proteus Providencia P. aeruginosaacinetobacter B. fragilis β E. coli P. aeruginosa

5 Methicillin-susceptible Staphylococcus aureus (MSSA) Methicillin-susceptible coagulase-negative staphylococci (MSCNS) Table3.Susceptibilities of clinical isolates to antimicrobial agents tested Drug MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST 284 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX Streptococcus pneumoniae 267 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX Penicillin-susceptible Streptococcus pneumoniae (PSSP) 125 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX (Continued) : Susceptibilities with breakpoint of the susceptible-dose dependent interpretive category.

6 Penicillin-intermediate resistant Streptococcus pneumoniae (PISP) Penicillin-resistant Streptococcus pneumoniae (PRSP) Streptococcus species (other than S. pneumoniae) Drug Table3.(Continued) MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST 84 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX Enterococcus faecalis 197 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX : Susceptibilities with breakpoint of the susceptible-dose dependent interpretive category. (Continued)

7 Drug MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST Moraxella catarrhalis 202 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX Escherichia coli 290 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM (91.0) 81.4 IPM MEPM GM CPFX LVFX ESBLs-producing Escherichia coli Table3.(Continued) 55 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM (52.7) 3.6 IPM MEPM GM CPFX LVFX Citrobacter species 243 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM (91.8) 86.0 IPM MEPM GM CPFX LVFX Klebsiella pneumoniae 207 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM (96.6) 92.8 IPM MEPM GM CPFX LVFX : Susceptibilities with breakpoint of the susceptible-dose dependent interpretive category. (Continued)

8 Drug MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST Enterobacter cloacae 168 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM (98.2) 83.3 IPM MEPM GM CPFX LVFX Serratia marcescens 250 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM (100) 98.0 IPM MEPM GM CPFX LVFX Proteus mirabilis 219 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM (97.7) 93.6 IPM MEPM GM CPFX LVFX Indole-positive Proteus species Table3.(Continued) 118 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM (100) 100 IPM MEPM GM CPFX LVFX Providencia species 66 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM (100) 97.0 IPM MEPM GM CPFX LVFX : Susceptibilities with breakpoint of the susceptible-dose dependent interpretive category. (Continued)

9 Drug MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST Haemophilus influenzae 265 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX lactamase-negative ampicillin-susceptible Haemophilus influenzae (BLNAS) -lactamase-negative ampicillin-resistant Haemophilus influenzae (BLNAR) Table3.(Continued) 102 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM EM CPFX LVFX Pseudomonas aeruginosa 286 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM CPFX LVFX : Susceptibilities with breakpoint of the susceptible-dose dependent interpretive category. (Continued)

10 Drug Table3.(Continued) MIC: g/ml Susceptibilities (%) MIC range MIC50 MIC80 MIC90 CLSI EUCAST Acinetobacter species 249 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM CPFX LVFX Bacteroides fragilis group 163 TAZ/PIPC PIPC SBT/ABPC SBT/CPZ CAZ CFPM IPM MEPM GM CPFX LVFX : Susceptibilities with breakpoint of the susceptible-dose dependent interpretive category. TAZ/PIPC: tazobactam/piperacillin, PIPC: piperacillin, SBT/ABPC: sulbactam/ampicillin, SBT/CPZ: sulbactam/cefoperazone, CAZ: ceftazidime, CFPM: cefepime, IPM: imipenem, MEPM: meropenem, GM: gentamicin, CPFX: ciprofloxacin, LVFX: levofloxacin, EM: erythromycin CLSI: Clinical and Laboratory Standards Institute, EUCAST: European Committee on Antimicrobial Susceptibility testing Acinetobacter E. cloacae S. marcescens β S. pneumoniae E. faecalis M. catarrhalis μ E. coli E. coli E. coli Citrobacter K. pneumoniae E. cloacae S. marcescens P. mirabilis Proteus Providencia

11 H. influenzae β Haemophilus influenzaeβ β Haemophilus influenzaeβ P. aeruginosa Acinetobacter Bacteroides fragilis III β β E. faecalis M. catarrhalise. colicitrobacter K. pneumoniaee. cloacaes. marcescens Proteus Providencia P. aeruginosaacinetobacter B. fragilis β β β β E. coli K. pneumoniae β β P. aeruginosa Acinetobacter E. cloacae S marcescens P. aeruginosa S. marcescens β E. colik. pneumoniae P. mirabilis β

12 β β β Escherichia coli Enterobacteriaceae Pseudomonas aeruginosa

13 β β Moraxella catarrhalis Escherichia coli Citrobacter Klebsiella pneumoniae Enterobacter cloacae Serratia marcescens Proteus Providencia Pseudomonas aeruginosa Acinetobacter Bacteroides fragilis β E. coli, K. pneumoniae P. mirabilis β P. aeruginosa Acinetobacter E. cloacae S. marcescens E.cloacae S. aureus M. catarrhalis P. mirabilis Proteus H. influenzae β

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